Bophelo, Litokisetso
Efferalgan - litaelo tsa tšebeliso
"Efferalgan" - e antipyretic ratoang. Le sebopeho lona ke batlang a fapane hanyenyane ho itšetlehile ka mofuta o lokolloe. Sebopeho sa sirapo bana - paracetamol le dikarolo ea thusang: sirapo, saccharin, nhua polyethylene glycol, E202, flavors, acid e citric, metsi a nwehang.
Standard fumaneha ka vials khalase ka etsang dilitara 0.09 (ka ho eketsehileng - lekanyang khaba).
Sebopeho "Efferalgan" (rectal): paracetamol, malandi ke seka-acylglycerol.
Standard ka dipalokatisanetswa likotoana 5, 'me ka pakete e ho na le 2 ambalaji.
Ka ho hlophisoa ha effervescent matlapa paracetamol le dikarolo ea thusang: omileng sodium carbonate, povidone, acid e citric, saccharin, sorbitol, sodium docusate, ho baka soda le ho e, E211.
Lipoleiti tse matlapeng a 4, le sephutheloana kaofela - ho na le 4, o na direkoto tsa 25.
litla diokobatsi
"Efferalgan" pukwanana hlalosa lithethefatsi, tse khōlō a sebetsang a ntho e paracetamol, eo ho na le masakana cyclooxygenase-1 le ea 2 haholo-holo ka ho CNS, kahoo ikitlaetsa tšusumetso e ka likoloha thermoregulatory le bohloko. Ka lisele tse fubileng ketso ea paracetamol ka Cox thibetsoeng khethehileng, peroxidases itseng. Sena ke seo e hlalosa ho ba sieo ha hoo e ka bang ka ho feletseng dintho-ba khahlanong le a hlabang a sebetsang. Paracetamol hase ka tsela efe kapa efe ama sebopeho sa prostaglandins ka lisele pheriferale, e hlalosang ho hloleha ka ho feletseng ho susumetsa mucosa gastrointestinal le ho leka-lekana electrolyte-metsi.
Likerese "Efferalgan" taeo e hlahisang bobeli moemeli le analgesic, antiinflammatory le antipyretic unexpressed sebediswa.
Paracetamol hangata ho thuisoa ho feletseng 'me ka potlako. Ea mahloriso palo e kahodimodimo ea lithethefatsi ka serum ka le hlaha ka mor'a metsotso 30-60. ka mor'a ho noa joala. Ka potlako ajoa ho pholletsa le lisele tsa mmele, paracetamol e hampe tlameha ho liprotheine lero la mali (ho fihlela ho 25%). O kenella ka hare ho ea mali-boko mokoallo.
Sam metabolism hlahisoang ke sebete. Paracetamol ke khumo le 'mele e le metabolites. E bontšoa ka mokgwa o ka sehloohong oa% 5 feela ea thero ea.
ya litatoli na
Lithethefatsi "Efferalgan" tataiso e khothalletsa maemo latelang le mafu a:
- bobeli antipyretic lithethefatsi tlas'a tloaelehileng OCR pathologies tšoaetsanoang bongoaneng, ntaramane, mathata postprivivochnyh, mafu a tšoaetsanoang le a hlabang tse tšoauoa ka hyperthermia;
- jwalo ka analgesic bakeng sa ka tsela e itekanetseng le ba fokolang bohloko (hlooho e opang, bohloko ka mesifa striated, meno bohloko, pheriferale diso methapo ea kutlo, bohloko ka chesa le ho sithabela).
Contraindications
Contraindications ea ho fumana 'Efferalgan "thuto e bontša joalo (kerese, sirapo)
- ditlolo ka lintho tse tebileng dithulaganyo tsa sebete kapa a liphio;
- eketseha susceptibility ho motsoako ka sehloohong;
- lefu ea mali;
- lilemo la khoeli e 'ngoe (bakeng sa sirapo) le ho fihlela ho likhoeli tse tharo (bakeng sa suppositories 0,08 g);
- haelloa ke potlakisang tsebetso ea lik'hemik'hale G-6-PD;
- mali kapa likarabo hlabang ka rectum (suppository).
Nkiloeng ka hloko lithethefatsi lokela ho ba:
- ka ho hloleha e amanang le sebete le renal (ke hore, ha cholehemia lelapa);
- ka renal ho hloleha bonyane lekhalo pakeng tsa ho sebelisa ho lokisetsa ho ka sirapo - lihora tse 8.
- sa kgothaletswa ho sebelisa likerese tsa letšollo.
Tablets "Efferalgan" taeo pukwanana ha ho kgothaletsa ka:
- eketseha susceptibility ho dikarolo;
- kamehla (khafetsa) tšebeliso ea joala;
- Boimana (1 le 3 trimesters) le nakong ea fepa ka;
- haelloa ke potlakisang tsebetso ea lik'hemik'hale G-6-PD;
- pele ka ba lilemo li leshome le metso e mehlano ( 'mele boima - ka tlase ho 50 kg) e.
Tablets le nkile ka hlokolosi:
- mafu ea sebete 'me liphio mosebetsi;
- ka congenital nyooko (Dubin-Johnson lefu, la lelapa cholehemia), lefu la sebete bongata ba kokwanahloko, ea lilemo li khōlō ho feta 60 a etsang dilitara tse, lefu sebete (joala) ..
litla-morao
Le litla-morao ha ho nka "Efferalgan" Taeo lintlha-khōlō tsa tsona ke tsena:
- ka seoelo haholo - ho hlatsa, ho nyekoa ke pelo, allergy (lekhopho, urticaria, pruritus, angioedema);
- ipiletsa bohata ho ithusa hanngoe le deurinatsii;
- ho ruruha ea lera la mucous tsa rectum ea;
- ka seoelo haholo - thrombocytopenia, khaello ea mali, mali a fetang methaemoglobin ka khaello ea mali ea neutrophils leykotsitopeniya.
Haeba nako e telele kalafo ka bongata ka tsela e feteletseng e ka 'na hanyenyane nang le chefo e ho sebete' me liphio.
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