BopheloLitokisetso

"Tenorik": ulasan pelanggan tsa lingaka. Matlapa a eketsehileng khatello ea

Atleha haeba e joalo e ea lithethefatsi, e le "Tenorik"? Hlahloba lithethefatsi lena le ka siea e mong. Ka puisano e joalo le lingaka le bakuli ba ka ba bonolo ho etsa qeto ea kamoo moriana o ile a re, hore na e etsa hore liphetoho lehlakoreng le hore na ho sebetsana le mosebetsi oo.

A sehloohong sena a re hlalosa ka ho qaqileng thepa le litšobotsi "Tenorik" lithethefatsi. Hlahloba mamello nka liodara ngaka ea hae, o tla boela ho be le hanyenyane tlaase.

Sebopeho, sebopeho, tlhaloso, ambalaji

Ho lokisetsa "Tenorik" (100, 50 mg,) e marketed e tšoeu matlapa chitja le biconvex sebopeho le mola khefu.

Sebōpeho sa meriana ena e na le tse peli tse metsoako a sebetsang a: chlorthalidone le atenolol. Hape, paakanyong ena e na le metsoako e eketsehileng tse fanoang ka sebōpeho sa poone starch, sodium lauryl sulfate, lactose, polyvinylpyrrolidone, talc, silica, magnesium stearate le isopropanol.

Re ke ke ra bolela hore pilisi "Tenorik" (a tlhahlobo ka sesebelisoa sena, o ka bona qetellong ea sehlooho se reng,) ba koahetsoeng ka barbotage khethehileng filimi. Ho na le methylene chloride, isopropanol, talc, hypromellose, thaethaniamo dioxide, macrogol le oli vaseline.

Fumana nkoa e le ea lithethefatsi e ka ba ka dipakete blister kapa hlobolisa matlapa 28 kapa 100.

Meriana meriana Products

ke eng lipilisi "Tenorik"? Litaelo bakeng sa ho sebelisoa (lithethefatsi theko hase phahameng haholo) o tlaleha hore hona motswako antihypertensive moemeli, eo e khona ho etsa hore nako e telele hypotensive sebediswa.

The bohlokwa ba tsamaiso ya lithethefatsi ka eona ka lebaka la ho nka khato ka ea likarolo 2, kapa ho ena le diuretic (chlorthalidone) le beta1-adrenergic blocker (atenolol).

thepa senotlolo

Bitsoa atenolol cardioselective beta1-blocker. E leng bokhoni ba khetha ya dintho le decreases le eketseha litekanyetso li behoa ea moriana. Atenol ha e na lera ka hare e tiileng le litla sympathomimetic. Feela joaloka tse ling tse beta-blockers, e na le liphello tse mpe inotropic le haholo, ae fokotsang lebelo ho otla ha pelo.

Ha e le chlorthalidone, ke diuretic (sulfonamide netiazidny). Ho kgothaletsa tlhopho ya likarolo tse kang chlorine le sodium. Hape karolo ena eketsa secretion ea bicarbonate, magnesium le potassium. Molao-motheo oa bohato lona antihypertensive e amanang le excretion sodium.

Atenolol hammoho le oa diuretics ke molemo ho feta ho sebelisoa ha e mong le e ea likarolo tsena ka thoko.

Action nkoa e le ea lithethefatsi e ho hlokomelwa ho pholletsa le letsatsi (ka mor'a lethal dose e le ba se nang balekane ka litekanyetso li behoa ea letsatsi le letsatsi).

The kinetics ya moriana

Hobane lithethefatsi "Tenorik" analogs, theko ea tse bontšitsoeng tlaase mona, ke mokhoa kopantswe nahana ka thepa kinetic ea e mong le ya dintho le a sebetsang a ka thoko.

Atenolol e ananelang 40-50% pampitšaneng gastrointestinal. mahloriso lona lebetsoeng le e ile ea fihla ka mor'a lihora tse 4 ka mor'a a e-ja a Letlapa. Ho buisana le liprotheine ke hoo e ka bang 8-16%.

Atenolol e sa kopana le khanyang metabolism bontšitsoeng ka sebete. About 90% ya dintho e ananelang excreted sa fetohe bakeng sa lihora tse 8-9. nako ena ka 'na ba eketseha ka ho hloleha matla renal, kaha tlosa atenolol etsoa ke liphio.

Ha e le chlorthalidone, ke 60% ananelang pampitšaneng gastrointestinal. The lero la mali mahloriso e ile ea fihla lebetsoeng le eona ka mor'a lihora tse 12. Ho buisana le liprotheine tse ka bang 75%.

Chlorthalidone di behilwe ke liphio ka hare ho lihora tse 50.

ho bonahala

Ho tswa ho nkoa lithethefatsi eketsehileng khatello ea ho thusa hantle haholo. Ha e le hantle, ea bohlokoa kgatelelo ya madi, 'me ke tse khōlō,' me mohlomong e le pontšo feela ho sebelisoa.

Contraindications

Hona joale, u tseba, morero ofe ka abeloa "Tenorik" matlapa (bontšang bakeng sa moriana ona li ne li fanoa ka holimo). Empa, ka bomalimabe, ho na le ho nkoa e le a lithethefatsi le e lethathamo tsotehang tsa contraindications. E sa kgothaletswa ho nka ka:

  • cardiogenic makala;
  • pheochromocytoma;
  • bradycardia (a bontša sethoathoa);
  • mafu a le khōlō ajoa pheriferale;
  • hypotension (a hatela pele ho matla);
  • metaboliki acidosis;
  • Av-thibela likepe 1st le lengolo la 3rd;
  • SSS;
  • asma tsoelang pele;
  • pelo ea ho hloleha (bobeli a hlobaetsang le a sa foleng);
  • lefu la tsoekere;
  • vasospastic angina (Prinzmetal o angina);
  • gout;
  • obstructive la bronchitis;
  • hlobaetsang lefu la sebete;
  • hypoglycemia;
  • renal ho hloleha ho mofuta o hlobaetsang;
  • tlaase ho lilemo tse lilemo tse 18;
  • myasthenia gravis;
  • hypersensitivity ho metsoako ea meriana.

Mokhoa oa ho nka "Tenorik" khatello ea mali e phahameng?

bakuli ba batho ba baholo etellang lithethefatsi mahareng sa kgothaletswa litekanyetso li behoa ea 100 mg,. The lethal dose ea pele ea lithethefatsi e lokela ho ba 50 mg, hang ka letsatsi.

Ha e le batho ba hōlileng, ba lithethefatsi "Tenorik" ba abetsoe ho ngata e esita le tse nyenyane.

Bakuli ba nang le tshebedisano phytoteratology renal ke tse lakatsehang ho fokotsa maqhubu a ea etellang lipilisi.

E lokela ho ile a hlokomela hore ka mor'a hore tshebediso ya nako e telele tsebeliso ea lithethefatsi le tlas'a review, khanselwa lona Ho hlokahala hore a phethe butle-butle.

litla-morao

Baeti ba fihlelang ho "Tenorik" Tablets e ka khopisang e latelang liphetoho lehlakoreng:

  • bradycardia, e ile ea eketseha pelo hloleha, lipheletsong batang, orthostatic hypotension, arrhythmia, Av-ea le literata, matšoao a claudication hill, lefu Raynaud ya ;
  • pherekano, lethargy, hlooho e opang, lipono, psychosis hlobaetsang, paresthesia, feto-fetoha, ho tsekela, mokhathala, lefu la ho hlobaela, disorientation, thothofatsang Pono;
  • ommeng molomo, e ile ea eketseha sebete transaminases, mafu gastrointestinal, hepatotoxicity le cholestasis intrahepatic, pancreatitis, ho nyekoa ke pelo, pipitlelano, ho ipolaisa tlala;
  • leukopenia, purpura, thrombocytopenia, eosinophilia, agranulocytosis;
  • alopecia, liphetoho psoriasiform, leihlo omileng, exacerbation ea psoriasis, photosensitivity, rashes letlalo;
  • bronchospasm, hyperuricemia, hypokalemia, hyponatremia;
  • phytoteratology tsoekere mamello, ho eketseha ha palo ea lisireletsi antinuclear, fokotswa potency.

liphello tsena lehlakoreng ke ka seoelo ebile o bonolo.

analogues theko

matlapa a theko "Tenorik" ke 110-120 li-ruble. Ba ile ba ka nka sebaka sa lithethefatsi tse kang "Atenol", "Dinorik" kapa "Tenoret".

Reviews of moriana "Tenorik"

Hlahloba ho atleha ha sesebelisoa sena se ka siea e mong. Ho latela bakuli le lingaka, melemo ya sehlooho oa sesebelisoa sena ke tsena:

  • katleho;
  • theko e tlase.

The go tlhoka mesola ya lithethefatsi ena e kenyeletsa:

  • monyetla oa ho lahleheloa ke moriri le ntshetsopele ya ho hloka matla (tlhokomelo tsa nako e telele);
  • kgonego ya ketsahalo ea sethoathoa.

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