Bophelo, Litokisetso
"Phenylbutazone" (matlapa): litaelo bakeng sa ho sebelisoa, analogues, theko le ulasan pelanggan
From seo le kamoo ho ka sebelisa e balletsweng ke meriana "Phenylbutazone" (matlapa)? Litaelo bakeng sa ho sebelisoa, ho bonahala, thepa le lintho tse khethollang moriana tla tšohloa sehloohong sena.
Hape ho na le u tla fumana boitsebiso bo mabapi le kamoo ho fana, o ile a re ho bolela seo metsoako li kenyelelitsoe sebopeho lona (mafolofolo le ba khathetseng moeeng), 'me haeba a ena le litla-morao.
Metsoako le ambalaji tsa meriana
ke metsoako e leng ka lithethefatsi "Phenylbutazone" ke efe? Tablets di na le dipegelo ba mafolofolo motsoako o kang phenylbutazone. Hape lithethefatsi kenyeletsa: litapole starch, primelloza, magnesium stearate, sodium bicarbonate, talc le silica.
Lithethefatsi "Phenylbutazone" (matlapa) e rekiswa ho dipakete blister, tse kenyeleditsweng ka lebokoso ambalaji.
Pharmacodynamic litšobotsi tsa moriana
Na u ne u tseba hore ena ke lithethefatsi e le "Phenylbutazone"? profesionalce Reviews tlaleha hore ke batho bao e seng steroidal-ba khahlanong le a hlabang moemeli eo o antipyretic le analgesic sebediswa.
Ho atleha ha moemeli ena e amanang le matla a ho thibela metsoako mosebetsi oa cyclooxygenase. Ka lebaka la tshusumetso joalo, ae fokotsang lebelo le tswakana tsa prostaglandins.
O ne a nka moriana o kgothaletsa ho reabsorption ea letsoai le metsi ho tubules le renal. E boetse e felisa bohloko le ho fokotsa ho ruruha, eo e atisa ho tsamaisana le ho ruruha.
Joang phello phekolo "Phenylbutazone" lithethefatsi? Tablets fokotsa bohloko kopanetsoeng (nakong tshisinyo le phomotse), hammoho le tsamaiso kapa keketseho ea bona fokotswa fapaneng ya tshisinyo.
-Ba khahlanong le a hlabang bohato ba moemeli ena ke haholo-holo phahametse "Amidopyrine" tšoanang lithethefatsi.
Ha gout a sebetsang a moriana o habeli urate excretion ka moroto, 'me ho fokotsa palo ea mali.
Hape hlokomela hore lithethefatsi "Phenylbutazone" (matlapa), litaelo bakeng sa tšebeliso eo e aa ageletsweng ka sephutheloana le machachetsi, ho fokotsa bohloko le ho ruruha le matšoao ha thrombophlebitis (postoperative le methapong hemorrhoidal).
Kinetic litšobotsi tsa ho lokisetsa ya
lithethefatsi "Phenylbutazone" (matlapa) moo ananelang? Motataisi o tlaleha hore absorption phahameng ya moriana pampitšaneng gastrointestinal se hlahile. bioavailability lona e ka 87-90% le lebetsoeng le lero la mali mahloriso e ketekoa ka mor'a metsotso e 60-150 ka mor'a tsamaiso.
From mali lithethefatsi butle-butle e ntse e feta ka lisele tse le ho makala, 'me hape le kenella ka hare ka cavity kopanetsoeng le ka mali-boko mokoallo.
Metabolism tsa moemeli sena sebete. Ha a ntse a lona halofo bophelo bo lihora tse 19-25. Ke khumo ka liphio le moriana o ka pampitšana tshilong ya dijo.
Ho bonahala ho lozenges
Maemong a mang, ho laela le lithethefatsi "Phenylbutazone"? Tablets katleho bonahatsa bona ka bobona ka ho phekola:
- ankylosing spondylitis;
- tabanan;
- psoriatic ramatiki ;
- lupus le ramatiki;
- tenosynovitis le bursitis;
- gouty ramatiki ;
- algodismenorei;
- poso tshebedisano bohloko;
- leino le hlooho.
Hape, lithethefatsi ena e sebediswa bakeng sa ho imoloha ea boemong bo sa thabiseng ka neuralgia, sciatica, 'me chesa.
Contraindications ho fumana meriana
Ke bokae e rona nkoa e le ea lithethefatsi? theko lona ke eng? "Phenylbutazone" ka rekoa lebenkeleng efe kapa efe ea lithethefatsi bakeng sa theko ka theko e tlaase haholo. Re tla hlahisa e qetellong ea sehlooho se reng.
Na ho na le contraindications efe kapa efe ya meriana ee? Ho ea ka litaelo tseo, lithethefatsi ba ka 'na ha sebelisoa ha:
- tsoa mali ho tswa ho pampitšana gastrointestinal historing;
- mamellane ea acid e acetylsalicylic;
- pelo ea morethetho boloetse;
- hypersensitivity ho phenylbutazone;
- lesapo moko hatelloang;
- exacerbation ea ulcerative colitis le peptic seso lefu pampitšaneng ena tshilong ya dijo;
- decompensated pelo hloleha;
- e amanang le sebete le ho hloleha renal;
- hyperkalemia;
- tlaase ho lilemo tse lilemo tse 12;
- ho ima, haholo-holo trimesters pele le la boraro;
- ha noa meriana e meng e na le phenylbutazone.
Litaelo tsa tšebeliso "Phenylbutazone" lithethefatsi
Ho latela thuto e ho lokisetsa "Phenylbutazone" nkiloe ka molomo ka mor'a lijo 150 mg, makhetlo a mane ka letsatsi. The lethal dose phahameng ka ho fetisisa le 'ngoe ea moriana e 200 mg,,' me letsatsi le letsatsi - 600.
Ka nako ea phekolo le moemeli ena e itšetlehile ka le lefu lena le ho tiea tsa boemo ba mokuli. Lethal dose lekanang 400-600 mg, ka letsatsi, ka khona ho fokotsa palo ya moroto le lefu la tsoekere insipidus.
Bacha ba tloha ka ba lilemo 12 of pilisi "Phenylbutazone" thonya 75 mg, ka makhetlo a mararo ka letsatsi. Ho thibela le phello halefisang ea lithethefatsi ena ka mucosa la mala le e kgothaletswa ho noa lebese mofuthu.
Ka ho ba teng ha mafu articular le phello moriana o Amplified ke tsoa hong tsamaiso "prednisolone" (Infusion, i.v.).
Ho lokela ho hlokomeloe hore ho eketsa phekolo sephetho "Phenylbutazone" matlapa a kopana le mafura "Phenylbutazone".
liphetoho e bohloko ka mor'a a e-ja matlapa
Baeti ba fihlelang ho "Phenylbutazone" matlapa a ka etsa hore tse latelang liphetoho systemic:
- ho nyekoa ke pelo, bohloko ba ka mpeng, dyspepsia;
- ho hlatsa, aphthous stomatitis, lesokolla;
- ulceration tsa lera mucous tsa tshilong ya dijo pampitšana, letšollo, ringing litsebeng ea;
- gastrointestinal mali;
- gingival mali le hemorrhoids;
- phahameng khatello ea mali;
- itlhokomoloso sebeteng;
- tšoaroa ke hlooho, khaello ea mali, ho tepella maikutlo, leukopenia, ho tsekela;
- otsela, agranulocytosis, thabo, thrombocytopenia.
litla-morao ka mali le ho hloka discontinuation tsa kalafo lithethefatsi ho setsebi sa.
Sodium le tshegetsa le go tlotla metsi 'meleng tse amanang le ho nka "phenylbutazone" haholo sitisa le boemo ba bakuli ba le kgatelelo ya madi le CHF. motsotso ona hape hloka liphetoho kalafo.
lithethefatsi tšoanang le theko
"Phenylbutazone" matlapa (likotoana 20) ka rekoa bakeng sa 40-70 li-ruble.
Ha e le papiso e, ha ba ntse ba sebelisa mokhoa latelang: "Phenylbutazone-OBL", "Artrizin", "phenylbutazone", "Butalidon".
Reviews of bakuli ka meriana
Hona joale hore u tseba seo ha e lithethefatsi "Phenylbutazone" theko. matlapa a ba theko e tlaase, empa mabapi le recensioni, joale ba tla hlahisa mona ka tlase.
Hlahloba likarabo tsa bakuli ka lithethefatsi ena, re ka ka tsela e sireletsehileng etsa qeto ea hore e ka tsela e atlehang bontša ka boeona e ka tsohle utloa bohloko bo kopanetsoeng 'me mesifa. Empa, ho phaella ho ditshwaelo tsa tse molemo, bakuli ba hangata e etsa ho fihlela ho eena, 'me melaetsa negative. Ho ea ka bona, "Phenylbutazone" lipilisi hangata e baka mathata a sa gastrointestinal pampitsana le mali 'mele. Ntlheng ena, lingaka tse ngata ho kgothaletsa ho tlohela ho noa meriana ena, 'me nkela sebaka nang le koloi e sireletsehileng.
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