Bophelo bo botleLitokisetso

Biseptol: litaelo tsa tšebeliso

Sulfanilamidny lithethefatsi "Biseptol", thuto e tla be e behiloe ka tlase, ke mefuta e loketseng ea ho thibela likokoana-hloko bakeng sa batho ba nang le litlhaloso tse fapaneng bakeng sa kopo ea ho qetela.

Lebitso la khoebo la lithethefatsi ke Biseptol. Thupelo e na le lebitso la machaba: "Co-trimoxazole". Moriana ke setho se kopantsoeng sa likokoana-hloko, se akarelletsang karolelano ea 5: 1 ea sulfamethoxazole le trimethoprim.

Sulfamethoxazole, e sebetsang ka tsela e ts'oanang le para-aminobenzoic acid (PABA), e ama hampe tlhahiso ea acid e dihydrofolic lieleng tsa baktheria, e thibela ho kenella ha PABA molek'hule ea dihydrofolic acid. Trimethoprim e etsa ketso ea sulfamethoxazole, e thibela ho fokotseha ha dihydrofolic acid e le mofuta oa folic acid, tetrahydrofolic, e ikarabellang bakeng sa phapanyetsano ea protheine le ho ata ha sele e nyenyane. Kahoo, ka ho sebelisana ha likarolo tse peli tse thathamisitsoeng ka holimo, ho thehoa ha folic acid, e hlokahalang bakeng sa likokoanyana tse nyenyane bakeng sa ho qaptjoa ha metsoako ea purine, 'me ka mor'a moo ho na le nucleic acid (DNA le RNA), e hlōleha. Ka lebaka leo, ho thehoa ha liprotheine ho ferekane 'me lefu la libaktheria le hlaha.

Ka mokhoa oa ho itokisetsa "Biseptol" - ho emisoa, taelo ea tšebeliso, ho phaella ho lintho tse sebetsang, ho boetse ho bua ka lintho tse thusang: macroglagal glyceryl hydroxysitrate, magnesium aluminium silicate, carmellose sodium, citric acid, methylparahydroxybenzonate, sodium hydrogen phosphate, propyl parahydroxybenzonate, saccharinate ea sodium, maltitol, monko o monate Fragole, propylene glycol, metsi a hloekisitsoeng.

Ka mokhoa oa ho itokisa "Biseptol" - matlapa, thuto ea lintho tse thusang e akarelletsa starch ea litapole, talcum, magnesium stearate, polyvinyl joala, aseptins M le P, propylene glycol.

Tabeng ea ho lokisetsa "Biseptol" thuto e na le lintlha tse latelang:

Phekolo ea mafu a mafu a tšoaetsanoang le a chesang, a bakoang ke likokoana-hloko:

- mafu a tšoaetsanoang a pampiri ea ho hema;

- sinusitis, otitis media;

- Ho senyeha ha bokhoni, ho ba le meningitis;

- lisosa tse tšoaetsanoang tsa tsamaiso ea urogenital;

- Gonorrhea;

- mafu a tšoaetsanoang a tšoaetso ea lijo;

- Lisosa tse tšoaetsanoang tsa litlolo tse bonolo le letlalo.

Hape mabapi le tšebeliso ea lithethefatsi "Biseptol" thuto e na le boitsebiso bo latelang:

- 240 mg habeli ka letsatsi bakeng sa bana ba lilemo li 2-5;

- 480 mg habeli ka letsatsi bakeng sa bana ba lilemo li 6-12;

- 960 mg habeli ka letsatsi bakeng sa bana ba ka mor'a lilemo tse 12 le batho ba baholo.

Lithethefatsi li na le litla-morao tse bonolo, tse hlahang ka mor'a ho tlohela tšebeliso ea eona.

Litlhaloso tse amanang le tšebeliso ea lithethefatsi "Biseptol" taeo ke tse latelang:

- mafu a sebetsang sebeteng;

- mathata a sebetsang liphio;

- ho senya tsamaiso ea hematopoiesis;

- Ho fokola ha pelo;

- Ho haelloa ke li-glucose-6-phosphate dehydrogenase;

- Boimana;

- Nako ea ngoana e ka ba likhoeli tse tharo;

- ho ba teng ha hypersensitivity ho likarolo tsa eona.

Haeba mokuli a fumanoa a e-na le angina e bakoang ke streptococcus, morero oa lithethefatsi ena ha o bontšoe. E le ho qoba kristalllography, 'me ka lebaka leo, urolithiasis, ho hlokahala ho fana ka phepo e phahameng ea metsi. Ka tšebeliso ea nako e telele, ho hlahloba boemo ba mali ea mali ho hlokahala.

Ho amoheloa ha trimethoprim ka nako e le 'ngoe ho eketsa liketso tsa hypoglycemia - lihlahisoa tsa sulfonylurea.

Tšebelisano e kopanetsoeng ea thiazide diuretics e ka etsa hore mali a eketsehe haholoanyane le thrombocytopenia.

Lithethefatsi li eketsa ts'ebetsong ea ketso ea boipheliso ea phenytoin le phello ea warfarin anticoagulant.

U se ke ua sebelisa lithethefatsi tsena ka kakaretso le cyclosporine, lebaka la ho khethoa ke phetoho ea liphio, hobane boemo ba mokuli bo ka 'na ba senyeha.

Haeba ho feta tekano, ho hlokahala hore u hlakole lithethefatsi, hlatsoa mpa bakeng sa lihora tse 2, noa haholo, matla a diuresis, folinate ea calcium e laeloa.

Lithethefatsi li lethathamong la lithethefatsi tseo e leng lithethefatsi tsa bohlokoa le tsa bohlokoa.

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