Bophelo, Litokisetso
Naiz (Letlapa) - taeo e pukwanana.
foromo litekanyetso li behoa
ho lokisetsa e entsoeng ka mefuta e 3-lithethefatsi - fanyeha, matlapa dispersible le tloaelehileng. The ho fanyeha ke monko monate le keletso ea mosehla 'mala le tšobotsi haholo tatso ea lithethefatsi ena. ho fanyeha The ka redispersed ke sisinya ho vial.
Tablets di etsoa hoo e ka bang tse tšoeu, le o fokolang yellowish tinge. Matlapa a sebopeho chitja biconcave, bokaholimo lona bobeli ke le boreleli.
Nise sebopeho:
ho fanyeha
Active ntho
- Nimesulide - 50 mg, (5 di ml ho fanyeha)
Excipients:
- sorbitol
- tsoekere
- xanthan marenene
- propyl
- methylparaben
- asiti citric
- phaenapole tatso
- Yellow dae WS
- glycerol
- polysorbate
- metsi a hloekisitsoeng
matlapa dispersible
Active ntho
- Nimesulide - 50 mg, (Lethathamo 1).
excipients
- aspartame
- k'halsiamo phosphate
- microcrystalline selulose
- carboxymethyl starch
- starch poone
- talc
- magnesium stearate
- Colloidal silicon e dioxide e
- phaenapole tatso
matlapa
Active ntho
- Nimesulide - 100 mg, (Lethathamo 1).
Excipients:
- magnesium stearate
- K'halsiamo haedrojene phosphate
- microcrystalline selulose
- Anhydrous colloidal ka silicon
- starch poone
- Sodium starch glycolate
- hloekisitsoeng talc
The bohato diokobatsi ya moriana
bohato diokobatsi amana haholo-holo le Nise - lipilisi, ho rupela le na le ya data ya mefuta eohle litekanyetso li behoa. Lithethefatsi ke NSAID, e nang le ka ho sebopehong sulfonilidnuyu lona khomo. Nimesulide mohlomong amana inhibitors tsa Cox-2, e le hore e na le litla-ba khahlanong le a hlabang le analgesic, ho phaella moo, lithethefatsi fana ka litla analgesic, empa ka tekanyo e monyenyane.
The mochine ea nkang khato ea lithethefatsi amanang le hatelloang tsa tswakana tsa prostaglandins ka ho ruruha le tse hatelloang ya sebopeho sa radicals oksijene le thibelo ya myeloperoxidase ho lokolloa.
Pharmacokinetics
Nise ho phethahetseng ananelang pampitšaneng gastrointestinal, fihla lebetsoeng le lona maling se ka mor'a lihora tse 2. Lithethefatsi ke 99% protheine tlangwa.
Ho lokisetsa nize - matlapa tataiso eo e nkiloeng mehloling official, metabiliziruetsya ka sebete 'me excreted ka moroto, ka 98% ea lethal dose ea fumaneng ke khumo motšehare.
ya litatoli na
- mafu Rheumatic hore ntshetsa pele ka ntle ho komiki e kopanetsoeng
- tabanan
- Ho ruruha le bohloko ka mor'a ho buuoa
- Bohloko a bakoang ke dysmenorrhea
- Feberu le bohloko nakong hlobaetsang ruruha ka Lufthansa holimo
Ditlamorao tsa Nise
Tablets, ho rupela le ho eo hona joale e leng, e ka hlahisa lehlakore-litla ka tsamaiso ea tse fapa-fapaneng le ho makala:
Lehlakoreng liphello tsa ea lithethefatsi, e leng lebisa ho pampitšana tshilong ya dijo
- ho nyekoa ke pelo
- lesokolla
- bohloko mala
- tarry litulo
Le litla-morao tsa lithethefatsi, tse amanang le tsamaiso ea methapo e bohareng:
- hlooho
- otsela
- ho tsekela
Le litla-morao tsa lithethefatsi, e leng se amanang le kulisa:
- etymology
- lekhopho
- urticaria
litla tse ling lehlakoreng:
- Tshegetsa le go tlotla ka mokelikeli 'mele
- oliguria
- ho ruruha
contraindications Nise
E lethathamo la contraindications oo e kgothaletswa ho qoba ho nka lithethefatsi, 'me ha ho hlile ho hlokahala, feela rerisane ngaka ya hao.
- Tsoa mali ho tswa ho pampitšana gastrointestinal
- hloleha liphio
- e amanang le sebete ho hloleha
- Boimana le diabolololo
- Peptic lefu gastrointestinal
sebelisana lithethefatsi nize
Tablets, litaelo ka tšebeliso ea eo ha e fella ka ho ya data e feletseng le akaretsang ka ditshebeditsano tsohle lithethefatsi paakanyong ne tjena: sa kgothaletswa ka mahlahana a latelang - phenytoin, digoxin, diuretics efe kapa efe, lithethefatsi lithium, anticoagulants, lithethefatsi antihypertensive, NSAIDs, methotrexate, cyclosporin .
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