Bophelo, Litokisetso
Lithethefatsi "Spitomin": litaelo bakeng sa ho sebelisoa, ho bonahala, contraindications
Kajeno re u bolella mabapi le lithethefatsi ena, e le "Spitomin". Litaelo tsa tšebeliso, theko, recensioni, analogs le litšobotsi tsa lona - linako tsena tsohle na le thahasello bakuli hore ngaka e beuweng meriana ena. tlhahisoleseding tsohle tse hlokahalang ka fumanoa hamorao sehloohong sena.
Tlhaloso ea lithethefatsi, sebopeho lona, 'me ka bophara ambalaji
ke lithethefatsi "Spitomin" ke efe? Litaelo bakeng sa ho sebelisoa (o ile a hlalosa ho lokisetsa ho na e fanoa ka ho qaqa) pheha khang ea hore pilisi ena tšoeu odorless, sebopeho chitja le bataletseng, le chamfer le le Valium le fatiloeng «E151».
sesebelisoa sa na le buspirone hydrochloride le dikarolo ea thusang tse kang starch carboxymethyl, lactose monohydrate, magnesium stearate, sodium, microcrystalline selulose le colloidal anhydrous silica.
Ka rekisa lithethefatsi bo fihla ka dipakete blister le mabokose.
Molao-motheo oa ho sebetsa
Ke lintho life tse fumanehang bakeng sa lithethefatsi "Spitomin"? Litaelo bakeng sa ho sebelisoa (matlapa theko hlahiswa mona ka tlase) pheha khang ea hore moemeli ena anxiolytic, e amana le letoto la lihlooho tse bao e seng benzodiazepine 'me o na le phello antidepressant.
Ho fapana le anxiolytics a mang, lithethefatsi ena e na le se antiepileptic, sedative, hypnotic le thepa myorelaxant. Molao-motheo oa lona ho sebetsa e thehiloe liphellong tsa buspirone ka dopaminergic le serotonergic tsamaiso ea.
Hona ho bolela khetha thibela ho dopamine receptors (presynaptic) le eketsa lebelo la nyakallo ea methapo ea kutlo (dopamine) midbrain.
thepa life tse ling tse sa tlholeho ka lithethefatsi "Spitomin"? Litaelo bakeng sa ho sebelisoa e bolela hore Buspirone ke khetha leeme agonist ea 5-HT1A serotonin receptors. Ho ha e ame ho tlama ea receptors benzodiazepine le GABA, 'me ha ho ame psychomotor mosebetsi' me ha a etsa hore mamello. Ho phaella moo, ke sesebelisoa sena ha se potentiate phello ea lino tse tahang.
Phello phekolo ea lithethefatsi nkoa develops butle-butle le ho etsahala ka mor'a e 'ngoe kapa tse peli ka mor'a kalafo.
Kinetics ea chelete
Absorption ea lithethefatsi "Spitomin", litaelo bakeng sa tšebeliso eo e bontšitsoeng tlaase mona, le hlaha ka pampitšana ea gastrointestinal. Buspirone e pharaletseng metabolized nakong temana ka sebete. bioavailability lona ke 4% le lebetsoeng le lero la mali mahloriso e ile ea fihla ka mor'a hora e 'ngoe.
Buspirone Ho lokolloa hammoho le lebese. Ho fumana boitsebiso bo mabapi le ho kenella ka hare tsa moriana ka mokoallo placental haelloa.
Ho lokisetsa tsoa masi bakeng sa lihora tse hlano.
ya litatoli na
Le se laetsoeng "Spitomin" Letlapa? Litaelo bakeng sa ho sebelisoa e bontsha ho bonahala lintho tse latelang:
- autonomic ho se sebetse lefu;
- ho tšoenyeha ho hloka taolo ke generalized;
- a khaotsa ho tsuba syndrome, joala (jwalo ka phekolo adjuvant);
- tšoha boloetse ;
- mafu a tepelletsang (jwalo ka phekolo adjuvant).
Contraindications
Maemong a mang, ho e sa kgothaletswa ho sebelisa lipilisi "Spitomin"? Litaelo bakeng sa ho sebelisoa e re: pathologies latelang le maemo ao lethal dose ea meriana e contraindicated ka se:
- glaucoma;
- hypersensitivity ho metsoako ea moriana;
- myasthenia gravis;
- renal insufficiency, haholo;
- nyenyane lilemo;
- tsoa hong baeti ba fihlelang ho ea Mao inhibitors ;
- diabolololo;
- nakong ea bokhachane.
Le moemeli tlhokomelo e tsamaisoa ka sebete ho thatafala ha sebete le ho hloleha renal.
Moriana o "Spitomin": litaelo tsa tšebeliso
Analogs tsa lithethefatsi li tla hlahisa mona ka tlase.
Ea chelete ea ho ho nkoa ka ka nako e tšoanang ea letsatsi, pele kapa ka mor'a lijo.
moriana o thibetsoe ho sebelisa ka linako tse ling (ka ya tlhokeho) bakeng sa kalafo ya ho tšoenyeha, kaha phello ea oona ho phekola develops sebelisoa feela ka mor'a hore ka makhetlo-khetlo.
The litekanyetso li behoa ea meriana ena e khethiloeng le batho ka bomong. Ka tloaelo, ke 15 mg,. E lokela ho arotsoe ka tekanyetso 2-3.
The lebetsoeng le le 'ngoe lethal dose ke 30 mg, le palo e kahodimodimo ea letsatsi - 60 mg,.
Ka batho ba hōlileng ka eona e fetoloe ea lethal dose e hlokahala. Ha phytoteratology renal kapa e amanang le sebete moriana o lokela ho sebelisoa ka hloko ka tekanyetso e nyenyane.
litla-morao
Hangata meriana "Spitomin" hantle mameletse. Feela maemong a mang, ke sesebelisoa sena ke ditlolo itseng:
- sefubeng bohloko, ho robala ho hloka taolo, fainting, molikoalikoane, ho hypotension, hlooho e opang, kgatelelo ya madi;
- tšohile tšoenyeha, bokong ho potoloha ha mali mafu a, liphetoho dysphoric, decompensation ya ho hloleha pelo, e ile ea eketseha nahanela ho lerata, myocardial infarction, dysphoria, cardiomyopathy, nahana ho ipolaea, bradycardia;
- depersonalization, batang se mamellane, nyakallo, agoraphobia, hyperkinesis, tinnitus, ho tšoenyeha, ho hlohlona ka mahlong, lethargy, leihlo redness, lipono, ho Hoeleketsa, pherekano, mafu psychotic;
- thothofatsang pono, laryngitis, conjunctivitis, ho ruruha ya nasal mucosa, phytoteratology tatso, ho ba le boikutlo oa ntho e boima ka ho sefuba, mafu a kelello tsebe, hyperventilation, bohloko leihlo, ho hloka moea, photophobia, epistaxis, e ile ea eketseha khatello ea intraocular;
- galaktoreyu, ho nyekoa ke pelo, thyroid senya, flatulence, bosiu enuresis, ho ipolaisa tlala, takatso ea botona le koketsego ya, dysuria, salivation, mafu matsatsing, mali mala, ntsha peo lieha le tse ling.
Price, analogues, ulasan pelanggan
Litsenyehelo tsa ho ba moemeli ena ke ka bang 600 li-ruble. Haeba hlokahala, e nkeloa sebaka ke e analoge kang "Buspirone Sandoz."
Consumer ulasan pelanggan tsebisa hore lithethefatsi leo e le e ntle anxiolytic moemeli. Leha ho le joalo, ho ka nka feela setsebi mabapi le morero oa ka nako e telele (ha ka linako tse ling).
Similar articles
Trending Now