BopheloLitokisetso

"Betacam": litaelo bakeng sa ho sebelisoa, analogs le ulasan pelanggan

Ho felisa khatello e phahameng le ea mafu a sa tšoaneng cardiac sebelisa beta1 adrenoblokatornye ho bolela. meriana e mong joalo ke lithethefatsi "Betacam". Litaelo bakeng sa ho sebelisoa e mo hlalosa e le lithethefatsi tseo hlahisa cardioselective, antihypertensive le sympathomimetic bohato.

litšobotsi tse neng li tloaelehile

sesebelisoa sena ho nkoa a maiketsetso a beta1-adrenergic blocker. Hlahisoang ke Cyprus semela "Medokemi LTD" foromo Letlapa le tšoeu kapa haholo tšoeu barbotage selateng.

Moriana o "Betacam" taeo ka tlhaloso ya ba lokisetsa ho ea e na le mefuta e latelang: ba na le sebopeho lekaneng le bokaholimo biconvex, ho na le ho arola hlobolisa likotsi. Ha o roba letlapa, ka nako eo ho tla ba le litaba tse ka hare tsa ka hare tse tšoeu, kapa hoo e ka bang tse tšoeu.

Ka moriana o "Betacam" taeo ka tlhaloso moreki sephutheloana hlahisa tsela e latelang: pakete e mong e na le machachetsi tse tharo. E mong le e ea moeli poleiti seleng ea e tsa phutheloa ka matlapa a 10.

sebopeho

Ka moriana karolo ka sehloohong e ileng ea fuoa karolo jwale ka mokgwa wa betaxolol hydrochloride letsoai. The litekanyetso li behoa ea e mong le Letlapa ke 0,020 g,

A sebelisa "Betacam" taeo ka ho hlophisoa ha metsoako sa kopanele tšebeletsong o ile a hlalosa ntle mme bo hlalosang palo ea tsona. Tablets thehoa starchy sodium glycolate, tsoekere, lebese, magnesium stearate, microcrystalline selulose mofuta, aerosil, thaethaniamo oxide e, le nhua polyethylene glycol hydroxymethylpropylcellulose letšoao 400.

mochine oa bohato

Ka moriana "Betacam" taeo pukwanana tiisa cardioselective beta1 -adrenoblokatornuyu ntle sebōpeho sa motheo sa sympathomimetic mosebetsi se nang matla. Matlapa e bontša e fokolang ya lera botsitso katleho.

mosebetsi Antihypertensive ka lebaka la liketso tse fokotsa khumo cardiac tsa mesifa pelo le ho fokotsa le kutloelo-bohloko tlhotlheletso ka methapo ea mali le ho periphery ea.

Selectivity liphello tsa ea lithethefatsi ka sebopeho sa β 1 -adrenoreceptor ke ke bitsoa khetheng, hobane tekanyetso e phahameng ea betaxolol e ka ama β 2 receptor -adrenozavisimye sebopeho tse sebakeng lijana bronchi le mali.

Thibela ketso ya moriana, e kentse litšobotsi pharmacodynamic amanang le ea fokotseha ka lebelo leo pelo phomotse le nakong ea ho ikoetlisa. Ke ka lebaka la thibelo ea lihlopha β-adrenoceptor ka noute sinus, eo, ae fokotsang lebelo automaticity bona.

E boetse e ho fokotsa ho lokolloa ha myocardial hlollang le le boemong bo mafolofolo le etseng letho la 'mele, e leng e etsa hore ke antagonism tlhōlisano ea catecholamines le pheriferale methapo ea kutlo e qetellong ea mofuta adrenergic.

Lithethefatsi fokotsa systolic le diastolic khatello ea mali ka methapo ea phomotse le nakong ea ho ikoetlisa, ho fokotsa reflex orthostatic keketseho e ka maqhubu a ya pelehi pelo. Joalo le phello ea lithethefatsi e ho fokotsa mojaro ka myocardium ena.

Beta adrenoblokatornoe ho bolela le fana ka mosebetsi antihypertensive ke mochine latelang:

  • fokotseha khumo cardiac;
  • felisoa spasm ka mothapo ho ka periphery ho loketseng hore a nke khato e bohareng, e leng lekanyetsang ea pulse length le kutloelo-bohloko ho mabota vascular nakong braking mosebetsi renin.

Nako e telele tsamaiso ea lithethefatsi ha e fokotsa hypertension phello ea oona. Haeba re nka ka lethal dose ea se nang molekane betaxolol 0,005 kapa 0,04 g,, phokotsong khatello e tla bontša feela ka mor'a hore 3 kapa 4 hora.

Ka moriana, "Betacam" User Kopo e bontša hore taolo ya litekanyetso li behoa 0.005g sesosa antihypertensive le phello eo e matla e makhetlo a mabeli tlase ho feta ka letlapa eohle.

The lebetsoeng le antihypertensive mosebetsi oa mahloriso efe kapa efe ya betaxolol bonahala ka mor'a matsatsi a 7-14.

Phekolo dosages ea moriana o ha bakela ikemetseng cardiodepressivny e le hantle, ha ho na phello tsoekere metabolism, ho lieha ha eketsa cations sodium le mokelikeli ka lisele tse ka.

Seo e sebediswa

Lithethefatsi "Betacam" taeo ka bopaki kenyeletsang mela latelang:

  • phahameng khatello ea mali;
  • gogoga mothapo lefu myocardial mesifa hlollang, myocardium infarction ka tshebetso;
  • hypertrophic cardiomyopathy.

moriana e hlophisitsweng ha ho na le liphetoho tse ka pelo, tse boletsoe ka matsapa a sinus morethetho, tachyarrhythmias ventricular le mofuta supraventricular, lieha depolarization tsa myocardium e, arrhythmia amanang le prolapse ka belofo mitral, tlhahiso ka tsela e feteletseng ea li-hormone thyroid.

Mokhoa oa ho sebelisa

Ka moriana "Betacam" litaelo bakeng sa ho sebelisoa pente lethal dose ho itšetlehile ka boemo ba mokuli. All lethal dose seno letsatsi ka ho noa. Lijo ha e ame ho absorption ea meriana. Letlapeng lokela ho hlatsoa fatse le metsi a hloekileng.

Eketseha khatello ea mali tšoaroa letsatsi le letsatsi a simolla lethal dose ya ho tswa ho 0,005 ho 0,010 g, Ka mor'a matsatsi a 7 kapa ya 14, ha ho hlokahala, ho eketsa ka tjhelete e ya moriana o 0,020 g,

Ke mang ea sa lokelang ho sebelisa

Ha mong le e mong o dumella ho sebelisa mokhoa oa ho "Betacam" taeo pukwanana. Contraindications amanang le nahanela ka tsela e feteletseng ho le metsoako e, hammoho le betaxolol hydrochloride.

E sa ba laela hore bakuli ba na le sa foleng pelo mesifa insufficiency liforomo sinoatrialnuyu le atrioventricular blockage ka tekanyo bobeli le la boraro, bradycardia, hypotension, bronchial litlhaselo tsa asthmatic, itlelang feela angina.

Lithethefatsi "Betacam" matlapa litaelo bakeng sa ho sebelisoa a boela sa kgothaletswa mofuta seno le makala cardiogenic, vascular angiotrofonevroze qetellong, eketsa mesifa myocardial hlollang, asthenic ophthalmoplegia, endarteritis obliterans, emfizemnom lethopa ya dinama tse nyenyane tse ea matšoafo, a sa foleng obstructive la bronchitis tlhaku le lefu la tsoekere mellitus.

liphetoho tse totobetseng ka liphio le diso psoriatic e contraindicated bakeng sa kalafo ya.

liphetoho tse bohloko

litla bohloko le bolela "Betacam" dikopo User kenyeletsa lieha ho otla ha pelo, atrioventricular blockage, cardiac mesifa insufficiency, orthostatic a akhela khatello ea, mafutsana ajoa ka bophara periphery ea, matsoho hangata e batang le maoto, paresthesia. Kahoo sitisa tsamaiso e khopo vascular le pelo.

Bronchial spasm, lekhopho, urticaria, psoriasis, e omeletseng leihlo mucous lera e ka etsahala liphetoho lehlakoreng le matšoafo makala bonwang, letlalo.

Lithethefatsi ho ka etsa hore ho otsela, boemo asthenic, mafu a tepelletsang, mokhathala ka tsela e feteletseng, pherekano, matšoao a lipono, dizzy le hlooho e bohloko.

dithulaganyo rateheng tsamaisong ea silang lijo li amahanngoa le ho nyekoa ke pelo, retching, letšollo, ho lieha setulo cholestasis.

liponahatso tse ling tsa ketso ea lithethefatsi e ka ba fokotseha ea leukocyte le lisele tse platelet mali, 'me hape fokotseha potency.

Features ya kalafo

Amohela lithethefatsi leha e le efe e ka amanang le makolopetso a itseng, e leng se li itšetlehile ka lihlopha diokobatsi, ea ho hlophisoa le litekanyetso li behoa ea ea lithethefatsi a sebelisa.

Meriana "Betacam" taeo e tabeng ea ho sebelisa litaelo tse khethehileng ba fuoa bakeng sa e mong le e tabeng ea bao e seng maemo a, tse hlokang ho eloa hloko.

Kahoo, ka ho ba sethaleng sa pele sa kalafo le ka bakela ho hloka tsa mesifa pelo ka batho ba le tšekamelo ea ho kheloha ena.

Lipilisi "Betacam" masken matšoao a le boemong hypoglycemic, tseo boholo ba tsona e nkoa e le tlōlo ea morethetho cardiac. Tsebo ena e lokela ho ela bakuli akhaonteng ba phahameng mali tsoekere. Ba hlokang go baya leitlho ea kamehla ea maemo tsoekere mali.

Haeba u sebelisa lithethefatsi, "Betacam" (matlapa) taeo e pukwanana khothalletsa lefa a lebisa tlhokomelo ho laola lebelo leo pelo. Tabeng ea mafu a bradycardic sinus morethetho, e litekanyetso li behoa hlokahalang ho fokotsa kapa hlakola e moemeli ya data kalafo.

Ho hloka tšebeliso hloko moriana ka bakuli ba thuto pheochromocytoma.

The meriana hammoho le ho bolela hore inhalation thethebatso e atlehe, o baka ho tepella maikutlo ea myocardial hlollang le tshebetso mesifa le ho theola khatello ea mali. Bao e seng depolarizing relaxants mesifa bontša ka nako e telele matlapa bohato ha pepesehetse "Betacam".

Ha o batla ho phetha ka ho ne ho reriloe buoa kenella tlhaku, ho lokisetsa hlakola matsatsi a mabeli pele ho ketsahalo eo matlapa a ne ke sa ama e thethebatso kakaretso.

Moriana o setopong kalafo "Betacam" taeo pukwanana buella se hang, empa butle-butle, le ho fokotseha ha dosing bakeng sa matsatsi a 7 kapa ya 14, ho qoba ho itšoara joang ea phelang ho khanselwa lithethefatsi. Mong le e mong matsatsi a mararo palo ya moriana e fokotsehile ka 0,005 g,

Tablets ho nkoa le lithethefatsi tse retarders Monoamine dihydrobenzophenanthridine potlakisang tsebetso ea lik'hemik'hale.

bohato Hypotensive tsa lithethefatsi 'me fokotsa estrogen bananeng nonsteroidal antiinflammatory lithethefatsi tseo khina ho ions sodium le metsi, empa hape thibela metsoako e tswakana tsa metsoako prostaglandin ka liphio.

Tsoa hong tshebediso ya diltiazem, amiodarone, le verapamil lipilisi "Betacam" isang eketsehileng bohato inhibitory betaxolol hydrochloride ka myocardial hlollang le mesifa contractility le conductivity lona.

The meriana hammoho le lithethefatsi cardiac glycosidic khothalletsa atrioventricular le literata mofuta.

Hammoho le oa antihypertensives tse ling ho eketsa hypotensive mosebetsi matlapa "Betacam".

K'hok'heine fokotswa phekolo bohlokwa ba tsamaiso ea betaxolol ka tsamaiso bona tsoa hong.

Ha e kopana le "Betacam" matlapa agonists kapa xanthines etsa hore felloe bobeli ea mosebetsi oa bona.

Phenothiazines le betaxolol hydrochloride ke itšoara eketsa dikahare lona maling.

Medicine "Betacam" thibela litokisetso tlosa nang lidocaine kapa theophylline.

Sulfasalazine eketsa serum ea mahloriso ea betaxolol hydrochloride.

Ha ho na tlhahisoleseding e mabapi le ho sebelisoa ha lithethefatsi ho bakuli kokelo ea bana.

Temoso e hlokahalang ha a sebelisa matlapa ho batho ha u ntse khanna koloi, hammoho le basali ba baimana le lactating.

lisebelisoa tsena

Ke beta1-adrenoblokatornym lithethefatsi Administration go baya ka ditlhopha moriana "Betacam" taeo pukwanana. Analogs hape ho matleng a sehlopha sena sa pharmacotherapeutic. Ba na le ba mafolofolo ba motsoako o liketso e le betaxolol hydrochloride.

French e nkoa e le analoge ea lithethefatsi "Lokren", e hlahisoang ke "Sanofi Winthrop Industry" tse tlang e le letlapa tlotsitsoeng tšoeu filimi. Theha tsona ho potoloha ka lifahleho biconvex, eo ho eona kotsi e leng le arola balla tlotla "KE 20".

Ho na le ke lethal dose 'ngoe ea 0,02 g, ea betaxolol hydrochloride. Thusang dikarolo meriana kenyeletsa lebese tsoekere, microcrystalline selulose, sodium carboxymethyl mofuta A, colloidal silicon e dioxide, magnesium stearate.

Filimi barbotage sebopeho ka lemoha hypromellose, nhua polyethylene glycol letšoao 400, thaethaniamo dioxide.

Lithethefatsi rekiswa ho lebokoso dipakete le machachetsi a mabeli a matlapa a 14.

Sebelisoa moriana ho felisa khatello e phahameng ea mali, e boetse e ho kopantswe le lithethefatsi tse ling tse khahlanong le kgatelelo ya madi.

Lithethefatsi ka phetha mehato e thibelang ho bua le exacerbation ea angina ka foromo tsitsipana.

Russia tšoanang ho bolela ke lithethefatsi "Betaxolol", eo e hlahisoang ke "Moscow Endocrine semela" tse tlang e le matlapa a tšoeu filimi a tlotsitsoeng. Ba na le sebopeho potoloha ka lifahleho biconvex. The motsoako a sebetsang a ho nkoa betaxolol hydrochloride ka palo ea 0,020 g, le metsoako ea thusang kenyeletsa lebese tsoekere, sodium starch glycolate, dehydrated aerosil, magnesium stearate, microcrystalline selulose mofuta. barbotage filimi Ho thehoa ke polyvinyl joala dioxide e-thaethaniamo, talc, Macrogol 3350 cha, Opadry tšoeu-2.

sesebelisoa sena e sebediswa systemically le khatello e phahameng ea mali.

Ho na le meriana e mong "" Betaxolol "tse tlang e le marotholi a mahlo, tse sebelisoa ka lihlooho ka foleng bulehileng-angle glaucoma mofuta le intraocular khatello e phahameng, ho tsosolosa Pono mora tham mong bang laser trabekuloplasticheskogo kenella.

maikutlo a bakuli

About bolela "Betacam" litaelo bakeng sa ho sebelisoa ka liphello tse sa lakatseheng tsa ulasan pelanggan e kenyeletsa karolo ea "Bohloko itšoare". le matšoao ana a ka se hakaalo hore e ba teng ha ba sebelisa lithethefatsi.

Bakuli ba bangata ka utloile poeletsotlaleho ntle ka ho beta1-adrenoblokatornom bolela "Betacam" hore ka ho phethahetseng o tšoara kgatelelo ya madi le angina. Ha e le hantle nka matlapa hammoho lithethefatsi tse ling antihypertensive ka phekolo e rarahaneng hore ntlafatsa sebetsa ka bona.

kalafo poso kgutlang khatello ea mali ho tloaelehileng, eo haholo ntlafatsa bophelo ba mokuli.

Ho boetse ho na ulasan pelanggan ya lithethefatsi tse bontšang katleho ha ea phekolo le moemeli ena.

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